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Selective Receptor Modulators

Meaning

Selective Receptor Modulators (SRMs) are a class of synthetic compounds that exhibit tissue-specific agonistic (activating) or antagonistic (blocking) effects on a specific type of hormone receptor. These compounds are designed to elicit beneficial effects in target tissues, such as bone or muscle, while minimizing undesirable side effects in other tissues, such as the prostate or breast. They represent a significant advance in targeted hormone therapy.