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Hexarelin

Meaning

Hexarelin is a synthetic hexapeptide that functions as a potent, orally active Growth Hormone Secretagogue (GHS). It is designed to stimulate the release of endogenous growth hormone (GH) by acting on the ghrelin/GHS receptor, primarily in the pituitary gland and hypothalamus. Clinically, it has been studied for its potential effects on cardiac function, muscle growth, and GH deficiency, showcasing a unique profile of action compared to GHRH analogues. Its therapeutic application is rooted in leveraging the body’s natural GH release pathways.