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Estrogen Blockers

Meaning

Estrogen Blockers are a class of pharmacological agents designed to interfere with the biological activity of estrogen by either reducing its production or inhibiting its binding to cellular receptors. Clinically, these medications are primarily utilized in oncology to treat hormone-sensitive cancers, but they also have applications in managing conditions where estrogen excess contributes to pathological states, such as gynecomastia or certain aspects of hormonal imbalance. These agents work to re-establish a more favorable systemic hormone profile, making them a powerful tool in precision endocrinology for both men and women. They require careful clinical oversight due to their profound impact on the endocrine system.