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Bioavailability Profiling

Meaning

Bioavailability Profiling is a pharmacokinetics-based clinical assessment that determines the fraction of an administered hormone or compound that reaches the systemic circulation and is available to exert its intended biological effect. This evaluation is essential in personalized hormonal therapy, as it quantifies the true therapeutic exposure rather than merely the administered dose. Understanding a patient’s unique absorption and metabolism profile is critical for achieving precise therapeutic outcomes and minimizing potential side effects. It provides the necessary data to adjust dosage forms and routes of administration for optimal efficacy.